P5514-100G Display Image

Pyrilamine maleate salt,

Code: P5514-100G D2-231

Application

Pyrilamine maleate salt has been used:to treat Cassiopea sp. as H1 receptor antagonistto intraperitoneally inject mice to prevent the release ...


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Your Price
£277.00 100G
£332.40 inc. VAT

Application

Pyrilamine maleate salt has been used:to treat Cassiopea sp. as H1 receptor antagonistto intraperitoneally inject mice to prevent the release of endogenous histaminein membrane binding assay to determine the Ki values and in the comparative inhibitory concentration (IC50) studies by whole-cell patch clamp technique

Biochem/physiol Actions

Pyrilamine maleate is a H1 histamine receptor antagonist. Pyrilamine maleate induces sleep in vertebrates. In Cassiopea, it induces concentration dependent dormancy.

Features and Benefits

This compound was developed by Watson. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

This compound is featured on the Histamine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Packaging

5, 25, 100 g in glass bottle

formpowder
Gene Informationhuman ... HRH1(3269)
InChI keyJXYWFNAQESKDNC-BTJKTKAUSA-N
InChI1S/C17H23N3O.C4H4O4/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15;5-3(6)1-2-4(7)8/h4-11H,12-14H2,1-3H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
originatorWatson
Quality Level100
SMILES stringOC(=O)C=C/C(O)=O.COc1ccc(CN(CCN(C)C)c2ccccn2)cc1
Code
Description
Unit Size
List Price
Qty
P5514-25G
Unit:25G
List Price: £118.00
Source:List Price
ADD
P5514-5G
Unit:5G
List Price: £35.80
Source:List Price
ADD
Cas Number59-33-6
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