B2134-250MG Display Image

2-Bromo-alpha-ergocryptine methanesulfonate salt, solid

Code: B2134-250MG D2-231

Application

2-Bromo-α-ergocryptine methanesulfonate salt has been used:as D2 agonist in bird zebra finchesfor Prl secretion inhibitor in micefor the inhibition of motility in...


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£564.00 250MG
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Application

2-Bromo-α-ergocryptine methanesulfonate salt has been used:as D2 agonist in bird zebra finchesfor Prl secretion inhibitor in micefor the inhibition of motility in planaria worm

Biochem/physiol Actions

Bromocriptine is an ergot alkaloid and a dopamine D2 receptor agonist. It is prescribed for Parkinson′s disorder, hyperprolactinemia and galactorrhoea. It modulates β cells of the pancreas from insulin hypersecretion and improves the metabolic profile in type 2 diabetes patients with obesity. It also modulates glutamate release by glutamate transporter,GLT-1.

colorwhite
formsolid
Gene Informationhuman ... DRD2(1813), DRD3(1814), PRL(5617)
InChI keyNOJMTMIRQRDZMT-NEKRQHSLSA-N
InChI1S/C32H40BrN5O5.CH4O3S/c1-16(2)12-24-29(40)37-11-7-10-25(37)32(42)38(24)30(41)31(43-32,17(3)4)35-28(39)18-13-20-19-8-6-9-22-26(19)21(27(33)34-22)14-23(20)36(5)15-18;1-5(2,3)4/h6,8-9,13,16-18,23-25,34,42H,7,10-12,14-15H2,1-5H3,(H,35,39);1H3,(H,2,3,4)/t18?,23-,24+,25+,31-,32+;/m1./s1
optical activity[α]20/D +95°, c = 1 in methanol: methylene chloride (1:1)(lit.)
Quality Level100
SMILES stringCS(O)(=O)=O.[H][C@@]12Cc3c(Br)[nH]c4cccc(C1=CC(CN2C)C(=O)N[C@@]5(O[C@]6(O)N([C@@H](CC(C)C)C(=O)N7CCC[C@@]67[H])C5=O)C(C)C)c34
solubilityH2O: 0.8 mg/mL, ethanol: 23 mg/mL
storage temp.2-8°C
Code
Description
Unit Size
List Price
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B2134-100MG
2-Bromo-alpha-ergocryptine methanesulfonate salt, solid

Unit:100MG
List Price: £317.00
Source:List Price
ADD
B2134-25MG
2-Bromo-alpha-ergocryptine methanesulfonate salt, solid

Unit:25MG
List Price: £95.40
Source:List Price
ADD
Cas Number22260-51-1
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